Publikationen des BMWZ


  • Cox RJ, Wang C, Lambert C, Hauser M, Deuschmann A, Zeilinger C, Rottner K, Stradal T, Stadler M, Skellam E (2020): Diversely Functionalised Cytochalasins via Mutasynthesis and Semi-Synthesis. Chemistry
    DOI: 10.1002/chem.202002241
  • Cox RJ, Wang C, Lambert C, Hauser M, Deuschmann A, Zeilinger C, Rottner K, Stradal T, Stadler M, Skellam E (2020): Diversely Functionalised Cytochalasins via Mutasynthesis and Semi-Synthesis. Chemistry
    DOI: 10.1002/chem.202002241
  • Heard, David M., Tayler, Emyr R., Cox, Russell J., Simpson, Thomas J., Willis, Christine L. (2020): Structural and synthetic studies on maleic anhydride and related diacid natural productsTETRAHEDRON, 2020, 76
    DOI: 10.1016/j.tet.2019.130717
  • Lukas Kahlert, Eman F. Bassiony, Russell J. Cox and Elizabeth J. Skellam (2020): Diels Alder Reactions During the Biosynthesis of SorbicillinoidsAngewandte Chemie, 2020, in press
  • Marc Stadler, Christopher Lambert, Daniel Wibberg, Jörn Kalinowski, Russell J. Cox, Miroslav Kolařík, Eric Kuhnert (2020): Intragenomic polymorphisms in the ITS region of high quality genomes of the Hypoxylaceae (Xylariales, Ascomycota)Mycological Progress, 2020, in press
    DOI: 10.1007/s11557-019-01552-9
  • Verena Hantke, Elizabeth J. Skellam, Russell J. Cox (2020): Evidence for enzyme catalysed intramolecular [4+2] Diels–Alder cyclization during the biosynthesis of pyrichalasin H.Chemical Communications
  • Berndt, V.; Beckstette, M.; Volk, M.; Dersch, P.; Broenstrup, M. (2019): Metabolome and transciptome-wide effects of the carbon storage regulator A in enteropathogenic Escherichia coli.Scientific Reports 2019, 9
    DOI: 10.1038/s41598-018-36932
  • C. Greco, K. de Mattos-Shipley, A. M. Bailey, N. P. Mulholland, J. L. Vincent, C. L. Willis, R. J. Cox, T. J. Simpson (2019): Structure revision of cryptosporioptides and determination of the genetic basis for dimeric xanthone biosynthesis in fungiChem. Sci. 2019 in press
    DOI: 10.1039/c8sc05126g
    ISBN: 2930-2939
  • Hantke, Verena, Wang, Chongqing, Skellam, Elizabeth J., Cox, Russell J. (2019): Function of pathway specific regulators in the ACE1 and pyrichalasin H biosynthetic gene clustersRSC ADVANCES, 2019, 9
    DOI: 10.1039/c9ra07028a
    ISBN: 35797-35802
  • Hermane J, Eichner S, Mancuso L, Schröder B, Sasse F, Zeilinger C, Kirschning A (2019): New geldanamycin derivatives with anti Hsp properties by mutasynthesis. Org Biomol Chem. 17, 5269-5278
    DOI: 10.1039/c9ob00892f
  • Höhl M, Zeilinger C, Roth B, Meinhardt-Wollweber M, Morgner U (2019): Multivariate discrimination of heat shock proteins using a fiber optic Raman setup for in situ analysis of human perilymph. Rev Sci Instrum. 90, 043110
    DOI: 10.1063/1.5030301
  • Kniggendorf AK, Schmidt D, Roth B, Plettenburg O, Zeilinger C (2019): pH-Dependent Conformational Changes of KcsA Tetramer and Monomer Probed by Raman Spectroscopy. Int J Mol Sci., 20, pii: E2736
    DOI: 10.3390/ijms20112736
  • Krüger K, Reichel T, Zeilinger C (2019): Role of heat shock proteins 70/90 in exercise physiology, exercise immunology and their diagnostic potential in sports. J Appl Physiol. (1985), 126, 916-927
    DOI: 10.1152/japplphysiol.01052.2018
  • Lebe, Karen E., Cox, Russell J. (2019): O-Methylation steps during strobilurin and bolineol biosynthesisRSC ADVANCES, 2019, 9
    DOI: 10.1039/c9ra06412e
    ISBN: 31527-31531
  • Luebken, D.; Saxarra, M.; Kalesse, M. (2019): Tris(acetylacetonato) Iron (III): Recent Developments and Synthetic Applications.Synthesis-Stuttgart, 2019, 51(1), 161-177
    DOI: 10.1055/s-0037-1610393
  • Marchanka, A.; Carlomagno T. (2019): Solid-State NMR Spectroscopy of RNA.Methods Enzymol. 2019, 615, 333-371
    DOI: 10.1016/bs.mie.2018.08.029
  • Ozturk, I. Kutay, Dupont, Pierre-Yves, Chettri, Pranav, McDougal, Rebecca, Boehl, Ole J., Cox, Russell J., Bradshaw, Rosie E. (2019): Evolutionary relics dominate the small number of secondary metabolism genes in the hemibiotrophic fungus Dothistroma septosporumFUNGAL BIOLOGY, 2019, 123
    DOI: 10.1016/j.funbio.2019.02.006
    ISBN: 397-407
  • Szwalbe, A. J.; Williams, K.; Song, Z.; de Mattos-Shipley, K.; Vincent, J. L.; Bailey, A. M.; Willis, C. L.; Cox, R. J.; Simpson, T. J. (2019): Characterisation of the biosynthetic pathway to agnestins A and B reveals the reductive route to chrysophanol in fungi.Chemical Science 2019, 10(1), 233-238
    DOI: 10.1039/c8sc03778g
  • Ullah, S.; Seidel, K.; Tuerkkan, S.; Warwas, D. P.; Dubich, T.; Rohde, M.; Hauser, H.; Behrens, P.; Kirschning, A.; Koester, M.; et al. (2019): Macrophage entrapped silica coated superparamagnetic iron oxide particles for controlled drug release in a 3D cancer model.Journal of Controlled Release 2019, 294, 327-336
    DOI: 10.1016/j.jconrel.2018.12.040
  • Wang H, Stahl F, Scheper T, Steffens M, Warnecke A, Zeilinger C (2019): Microarray-based screening system identifies temperature-controlled activity of Connexin 26 that is distorted by mutations. Sci Rep. 9, 13543
    DOI: 10.1038/s41598-019-49423-3
  • Wang, Chongqing, Becker, Kevin, Pfuetze, Sebastian, Kuhnert, Eric, Stadler, Marc, Cox, Russell J., Skellam, Elizabeth (2019): Investigating the Function of Cryptic Cytochalasan Cytochrome P450 Monooxygenases Using Combinatorial BiosynthesisORGANIC LETTERS, 2019, 21
    DOI: 10.1021/acs.orglett.9b03372
    ISBN: 8756-8760
  • Wang, Chongqing, Hantke, Verena, Cox, Russell J., Skellam, Elizabeth (2019): Targeted Gene Inactivations Expose Silent Cytochalasans in Magnaporthe grisea NI980ORGANIC LETTERS, 2019, 21
    DOI: 10.1021/acs.orglett.9b01344
  • Warnecke A, Kirschning A, Landsberg D, Zeilinger C (2019): Hsp90: a target for susceptibilities and substitutions in biotechnological and medicinal application. Heat Shock Protein 90 in Human Diseases and Disorders, Ed Asea, Alexzander AA, Kaur, Punit (Eds.)
    DOI: 10.1007/978-3-030-23158-3
  • Warnecke A.; Kirschning A.; Landsberg D.; Zeilinger C. (2019): C Hsp90: a target for susceptibilities and substitutions in biotechnological and medicinal application.
  • Yang, Xiao-Long, Friedrich, Steffen, Yin, Sen, Piech, Oliver, Williams, Katherine, Simpson, Thomas J., Cox, Russell J. (2019): Molecular basis of methylation and chain-length programming in a fungal iterative highly reducing polyketide synthaseCHEMICAL SCIENCE, 2019, 10
    DOI: 10.1039/c9sc03173a
    ISBN: 8478-8489
  • Alizadeh H, Davoodi J, Zeilinger C, Rafii-Tabar H. (2018): Molecular dynamics simulation of the thermosensitivity of the human connexin 26 hemichannel, Chemical Physics, 500, 7–14
    DOI: 10.1016/j.chemphys.2017.11.002
  • Alizadeh, H.; Davoodi, J.; Zeilinger C.; Rafii-Tabar H. (2018): Molecular dynamics simulation of the thermosensitivity of the human connexin 26 hemichannelChemical Physics 2018, 500, 7-14
    DOI: 10.1016/j.chemphys.2017.11.002
  • de Mattos-Shipley, K. M. J.; Greco, C.; Heard, D. M.; Hough, G.; Mulholland, N. P.; Vincent, J. L.; Micklefield, J.; Simpson, T. J.; Willis, C. L.; Cox, R. J.; et al. (2018): The cycloaspeptides: Uncovering a new model for methylated nonribosomal peptide biosynthesis.Chemical Science 2018, 9(17), 4109-4117
    DOI: 10.1039/c8sc00717a
  • He Y., Wang B., Chen W., Cox R. J., He J. and Chen F. (2018): Recent advances in reconstruction microbial seconday metabolites biosynthesis in Aspergillus spp.Biotechnol. 36 (3), 2018 739-783
    DOI: 10.1016/j.biotechadv.2018.02.001
  • Kirschning, A.; Dibbert, N.; Draeger, G. (2018): Chemical Functionalization of Polysaccharides-Towards Biocompatible Hydrogels for Biomedical Applications.Chem-Eur. J. 2018, 24(6), 1231-1240
    DOI: 10.1002/chem.201701906
  • Kuhnert, E.; Li Y.; Lan, N.; Yue, Q.; Chen, L.; Cox, R. J.; An, Z.; Yokoyama, K.; Bills, G. F. (2018): Enfumafungin synthase represents a novel lineage of fungal triterpene cyclases.Environmental Microbiology 2018, 20(9,SI), 3325-3342
    DOI: 10.1111/1462-2920.14333
  • Lercher, L.; Danilenko, N.; Kirkpatrick, J.; Carlomagno, T. (2018): Structural characterization of the Asf1-Rtt109 interaction and its role in histone acetylation.Nucleic Acids Res 2018, 46(5), 2279-2289
    DOI: 10.1093/nar/gkx1283
  • Li, J.; Xing, J.; Luecke, D.; Luebken, D.; Millbrodt, L.; Plentz, R. R.; Kalesse, M. (2018): The Structure Elucidation of Haprolid.Synthesis-Stuttgart 2018, 50(3), 529-538
    DOI: 10.1055/s-0036-1591836
  • Luecke, D.; Linne, Y.; Hempel, K.; Kalesse, M. (2018): Total Synthesis of Pericoannosin A.Organic Letters 2018, 20(15), 4475-4477
    DOI: 10.1021/acs.orglett.8b01768
  • Marchanka, A.; Kreutz, C.; Carlomagno, T. (2018): Isotope labeling for studying RNA ba solid-state NMR spectroscopy.Journal of Biomolecular NMR 2018, 71(3,SI), 151-164
    DOI: 10.1007/s10858-018-0180-7
  • Marchanka, A.; Stanec, J.; Pintacuda, G.; Carlomagno, T. (2018): Rapid access to RNA resonances by proton-detected solid-state NMR at > 100 kHz MAS.Chemical Communications 2018, 54(65), 8972-8975
    DOI: 10.1039/c8cc04437f
  • Mattos-Shipley K., Lebe K. E., Han L.-C., Iqbal Z., Bailey A., Willis C., Simpson T. and Cox R. J. (2018): Strobilurin Biosynthesis in Basidiomycete FungiNature Commun. 9, 2018 3940
    DOI: 10.1038/s41467-018-06202-4
  • Mohammadi-Ostad-Kalayeh S, Stahl F, Scheper T, Kock K, Herrmann C, Batista FAH, Borges JC, Sasse F, Eichner S, Ongouta J, Zeilinger C, Kirschning A (2018): Heat shock proteins revisited using a mutasynthetically generated reblastatin library for comparing the inhibition of human with Leishmania Hsp90s. ChemBioChem, 19, 1–14
    DOI: 10.1002/cbic.201700616
  • Oberhauser, C.; Harms, V.; Seidel, K.; Schroeder, B.; Ekramzadeh, K.; Beutel, S.; Winkler, S.; Lauterbach, L.; Dickschat, J. S.; Kirschning, A. (2018): Exploiting the Synthetic Potential of Sesquiterpene Cyclases for Gnerating Unnatural Terpenoids.Angew. Chem. Int. Edit. 2018, 57(36), 11802-11806
    DOI: 10.1002/anie.201805526
  • Podrezova, E. V.; Larkina, M. S.; Belousov, M. V.; Kirschning, A.; Zhdankin, V. V.; Yusubov, M. S. (2018): Expedient Synthesis of Long-Chain omega-Substituted Fatty Acids and Esters from Cyclic Ketones using Iodine and Hydrogen Peroxide.Synthesis-Stuttgart 2018, 50(20), 4081-4088
    DOI: 10.1055/s-0036-1591598
  • Schmitt H, Roemer A, Zeilinger C, Salcher R, Durisin M, Staecker H, Lenarz T, Warnecke A. (2018): Heat Shock Proteins in Human Perilymph: Implications for Cochlear Implantation. Otol Neurotol. 39, 37-44
    DOI: 10.1097/MAO.0000000000001625
  • Schmitt, H.; Roemer, A.; Zeilinger, C.; Salcher, R.; Durisin, M.; Staecker, H.; Lenarz, T.; Warnecke, A. (2018): Heat Shock Proteins in Human Perilymph: Implications for Cochlear Implantation.Otology & Neurotology 2018, 39(1), 37-44
    DOI: 10.1097/MAO.0000000000001625
  • Schor, R.; Cox, R. J. (2018): Classic fungal natural products in the genomic age: the molecular legacy of Harold Raistrick.Nat. Prod. Rep. 2018, 35(3), 230-256
    DOI: 10.1039/c8np00021b
  • Schor, R.; Schotte, C.; Wibberd, D.; Kalinowski, J.; Cox, R. J. (2018): Three previously unrecognised classes of biosynthetic enzymes revealed during the production of xenovulene A.Nature Communications 2018, 9
    DOI: 10.1038/s41467-018-04364-9
  • Sommer, H.; Braun, M.; Schroeder, B.; Kirschning, A. (2018): 4-Ethoxy-1,1,1-trifluoro-3-buten-2-one (ETFBO), a Versatile Precursor for Trifluoromethyl-Substituted Heteroarenes - a Short Synthesis of Celebrex(R) (Celecoxib).Synlett 2018, 29(1), 121-125
    DOI: 10.1055/s-0036-1589097
  • Stempel, E.; Kaml, R. F.-X.; Budisa, N.; Kalesse, M. (2018): Painting argyrins blue: Negishi cross-coupling for synthesis of deep-blue tryptophan analogue beta-(1-azulenyl)-L-alanine and its incorporation into argyrin C.Bioorgan. Med. Chem. 2018, 26(19), 5259-5269
    DOI: 10.1016/j.bmc.2018.03.037
  • Surup, F.; Kuhnert, E.; Boehm, A.; Pendzialek, T.; Solga, D.; Wiebach, V.; Engler, H.; Berkessel, A.; Stadler, M.; Kalesse, M. (2018): The Rickiols: 20-, 22-, and 24-membered Macrolides from the Ascomycete Hypoxylon rickii.Chem-Eur. J. 2018, 24(9), 2200-2213
    DOI: 10.1002/chem.201704928
  • Yue Q, Stahl F, Plettenburg O, Kirschning A, Warnecke A, Zeilinger C (2018): The Noncompetitive Effect of Gambogic Acid Displaces Fluorescence-Labeled ATP but Requires ATP for Binding to Hsp90/HtpG. Biochemistry. 57, 2601-2605
    DOI: 10.1021/acs.biochem.8b00155
  • Yue, Q.; Stahl, F.; Plettenburg, O.; Kirschning, A.; Warnecke, A.; Zeilinger, C. (2018): The Noncompetitive Effect of Gambogic Acid Displaces Fluorescence-Labeled ATP but Requires ATP for Binding to Hsp90/HtpG.Biochemistry 2018, 57(18), 2601-2605
    DOI: 10.1021/acs.biochem,8b00155
  • Ammermann, J.; Schmidt, T.; Donner, J.; Reck, M.; Dalton, M.; Stumpp, N.; Stiesch, M.; Wagner-Doebler, I.; Kirschning, A. (2017): The carolactam strategy is ineffective: Synthesis and bioological evaluation of carolactam.Org. Biomol. Chem. 2017, 15(40), 8553-8558
    DOI: 10.1039/
  • Ceylan, S.; Law, H. C.-H.; Kirschning, A.; Toy, P. H. (2017): Organocatalytic Alkyne Isomerizations under Flow Conditions Using Heterogeneous Bifunctional Polystyrene Bearing Phosphine and Phenol Groups.Synthesis-Stuttgart 2017, 49(1), 145-150
    DOI: 10.1055/s-0036-1588589
  • Codutti, L.; Grimaldi, M.; Carlomagno, T. (2017): Structure-Based Design of Scaffolds Targeting PDE10A by INPHARMA-NMR.J. Chem. Inf. Model. 2017, 57 (6), 1488-1498
    DOI: 10.1021/acs.jcim.7b00246
  • Donner, J.; Reck, M.; Bunk, D.; Jarek, M.; App, C. B.; Meier-Kolthoff, J. P.; Overmann, J.; Mueller, R.; Kirschning, A.; Wagner-Doebler, I. (2017): The Biofilm Inhibitor Carolacton Enters Gram-Negative Cells: Studies Using a TolC-Deficient Strain of Escherichia coli.Msphere 2017, 2(5)
    DOI: 10.1128/mSphereDirect.00375-17
  • Essoung, F. R. E.; Mba'ning, B. M.; Mohamed, S. A.; Lwande, W.; Ngouela, S. A.; Tsamo, E.; Chhabra, S. C.; Hassanali, A.; Cox, R. J. (2017): Welwitschianalol A and B, two cyclohexene derivatives and other insecticidal constituents of Caesalpinia welwitschiana (Oliv.) Brenan.Phytochemistry Letters 2017, 22, 81-86
    DOI: 10.1016/j.phytol.2017.09.010
  • Feng, J.; Zhang, P.; Cui, Y.; Li, K.; Qiao, X.; Zhang, Y.-T.; Li, S.-M.; Cox, R. J.; Wu, B.; Ye, M.; et al. (2017): Regio- and Stereospecific O-Glycosylation of Phenolic Compounds Catalyzed by a Fungal Glycosyltransferase from Mucor hiemalis.Advanced Synthesis & Catalysis 2017, 359(6), 995-1006
    DOI: 10.1002/adsc.201601317
  • Gao, S.-S.; Wang, L.; Song, Z.; Hothersall, J.; Stevens, E. R.; Connolly, J.; Winn, P. J.; Cox, R. J.; Crump, M. P.; Race, P. R.; et al. (2017): Selected Mutations Reveal New Intermediates in the Biosynthesis of Mupirocin and the Thiomarinol Antibiotics.Angew. Chem. Int. Edit. 2017, 56(14), 3930-3934
    DOI: 10.1002/anie.201611590
  • Karaca, E.; Rodrigues, J. P. G. L. M.; Graziadei, A.; Bonvin, A. M. J. J.; Carlomagno, C. (2017): M3: an integrative framework for structure determination of molecular machinesNature Methods 2017, 14 897-902
    DOI: 10.1038/nmeth.4392
  • Kipke, A.; Schoening, K.-U.; Yusubov, M.; Kirschning, A. (2017): TEMPO-Mediated Oxidative Deformylation of Aldehydes: Applications in the Synthesis of Polyketide Fragments.Eur. J. Org. Chem. 2017, 46, 6906-6913
    DOI: 10.1002/ejoc.201701349
  • Liddle, E.; Scott, A.; Han, C.; Ivison, D.; Simpson, T. J.; Willis, C. L.; Cox, R. J. (2017): In vitro kinetic study of the squalestatin tetraketide synthase dehydratase reveals the stereochemical course of a fungal highly reducing polyketide synthase.Chemical Communications 2017, 53(10), 1727-1730
    DOI: 10.1039/c6cc10172k
  • Mohammadi-Ostad-Kalayeh S, Hrupins V, Helmsen S, Ahlbrecht A, Stahl F, Scheper T, Preller M, Surup F, Stadler M, Kirschning A, Zeilinger C (2017): Development of a microarray-based assay for efficient testing of new HSP70/DnaK inhibitors. Bioorg Med Chem, pii: S0968-0896(17), 31487-31486
    DOI: 10.1016/j.bmc.2017.10.003
  • Mohammadi-Ostad-Kalayeh, S.; Hrupins, V.; Helmsen, S.; Ahlbrecht, C.; Stahl, F.; Scheper, T.; Preller, M.; Surup, F.; Stadler, M.; Kirschning, A.; et al. (2017): Development of a microarray-based assay for efficient testing of new HSP70/DnaK inhibitors.Bioorgan. Med. Chem. 2017, 25(24), 6345-6352
    DOI: 10.1016/j.bmc.2017.10.003
  • Moore, B. S.; Carter, G. T.; Broenstrup, M. (2017): Editorial: Are natural products the solution to antimicrobial resistance?Nat. Prod. Rep. 2017, 34(7), 685-686
    DOI: 10.1039/c7np90026k
  • Poock, C.; Kalesse, M. (2017): Total Synthesis of Nannocystin Ax.Organic Letters 2017, 19(17), 4536-4539
    DOI: 10.1021/acs.orglett.7b02112
  • Roberts, D. M.; Bartel, C.; Scott, A.; Ivison, D.; Simpson, T. J.; Cox, R. J. (2017): Substrate selectivity of an isolated enoyl reductase catalytic domain from an iterative highly reducing fungal polyketide synthase reveals key components of programming.Chemical Science 2017, 8(2), 1116-1126
    DOI: 10.1039/c6sc03496a
  • Scherer, S.; Wollrab, E.; Codutti, L.; Carlomagno, T.; Gomes da Costa, S.; Volkmer, A.; Bronja, A.; Schmtz, O. J.; Ott, A. (2017): Chemical Analysis of a “Miller-Type” Complex Prebiotic BrothOrig. Life Evol. Biosph. 2017, 47 381-403
    DOI: /10.1007/s11084-016-9528-8
  • Seidel, K.; Balakrishnan, A.; Alexiou, C.; Janko, C.; Komoll, R.-M.; Wand, L.-L.; Kirschning, A.; Ott, M. (2017): Synthesis of Magnetic-Nanoparticle/Ansamitocin Conjugates-Inductive Heating Leads to Decreased Cell Proliferation In Vitro and Attenuation of Tumour Growth In Vivo.Chem-Eur. J. 2017, 23(50,SI), 12326-12337
    DOI: 10.1002/chem.201701491
  • Sharma R, Mohammadi-Ostad-Kalayeh S, Stahl F, Zeilinger C, Dräger G, Kirschning A, Ravikumar PC (2017): Two new labdane diterpenoids and one new β lactam compound from the aerial part of Roylea cinerea Phytochem. Lett, 19, 101–107
    DOI: 10.1016/j.phytol.2016.12.013
  • Sharma, R.; Mohammadi-Ostada-Kalayeh, S.; Stahl, F.; Zeilinger, C.; Draeger, G.; Kirschning, A.; Ravikumar, P. C. (2017): Two new labdane diterpenoids and one new beta-lactam from the aerial parts of Roylea cinerea.Phytochemistry Letters 2017, 19, 101-107
    DOI: 10.1016/j.phytol.2016.12.013
  • Trenti, F.; Cox, R. J. (2017): Structural Revision and Biosynthesis of the Fungal Phytotoxins Phyllostictines A and B.J. Nat. Prod. 2017, 80(5), 1235-1240
    DOI: 10.1021/acs.jnatprod.7b00183
  • W. Chen, R. Chen, Q. Liu, Y. He, K. He, X. Ding, L. Kang, X. Guo, N. Xie, Y. Zhou, Y. Lu, R. J. Cox, I. Molnar, M. Li, Y. Shao, F. Chen (2017): Orange, red, yellow: biosynthesis of azaphilone pigments in Monascus fungiChemical Science 2017
    DOI: 10.1039/c7sc00475c
  • Wang, L.-L.; Balakrishnan, A.; Bigall, N.-C.; Candito, D.; Miethe, J. F.; Seidel, K.; Xie, Y.; Ott, M.; Kirschning, A. (2017): A Bio-Chemosynthetic Approach to Superparamagnetic Iron Oxide-Ansamitocin Conjugates for use in Magnetic Drug Targeting.Chem-Eur. J. 2017, 23(10), 2265-2270
    DOI: 10.1002/chem.201604903
  • Wang, L.-L.; Candito, D.; Draeger, G.; Herrmann, J.; Mueller, R.; Kirschning, A. (2017): Harnessing a p-Quinone Methide Intermediate in the Biomimetic Total Synthesis of the Highly Active Antibiotic 20-Deoxy-Elansolid B1.Chem-Eur. J. 2017, 23(22), 5291-5298
    DOI: 10.1002/chem.201605884
  • Wang, L.-L.; Candito, D.; Draeger, G.; Kirschning, A. (2017): Synthetic Studies Probing Elansolid Biosynthesis: A para-Quinone-Methide-Triggered Intramolecular Diels-Alder Reaction.Eur. J. Org. Chem. 2017, 37, 5582-5591
    DOI: 10.1002/ejoc.201701125
  • Wang, L.-L.; Kirschning, A. (2017): Total synthesis of elansolids B1 and B2.Beilstein Journal of Organic Chemistry 2017, 13, 1280-1287
    DOI: 10.3762/bjoc.13.124
  • Williams K., Szwalbe A. J., Dickson C., Desson T. R., Mulholland N. P., Vincent J. L., Clough J. M., Bailey A. M., Butts C. P., Willis C. L., Simpson T. J., Cox R. J. (2017): Genetic and Chemical Characterisation of the Cornexistin Pathway Provides Further Insight into Maleidride BiosynthesisChem. Commun, 2017, in press
    DOI: 10.1039/C7CC03303F
  • Witte, S. N. R.; Hug, J. J.; Geraldy, M. N. E.; Mueller, R.; Kalesse, M. (2017): Biosynthesis and Total Synthesis of Pyrronazol B: a Secondary Metabolite from Nannocystis pusilla.Chem. Eur. J. 2017, 23(63), 15917-15921
    DOI: 10.1002/chem.201703782
  • Yusubov, M. S.; Postnikov, P. S.; Yusubova, R. Y.; Yoshimura, A.; Juerjens, G.; Kirschning, A.; Zhdankin, V. V. (2017): 2-Iodoxybenzoic Acid Tosylates: The Alternative to Dess-Martin Periodiane Oxidizing Reagents.Advanced Synthesis & Catalysis 2017, 359(18), 3207-3216
    DOI: 10.1002/adsc.201700776
  • Bowman, A.; Lercher, L.; Singh, H. R.; Zinne, D.; Timinszky, G.; Carlomagno, T.; Ladurner, A. G. (2016): The histone chaperone sNASP binds a conserved peptide motif within the globular core of histone H3 through its TPR repeats.Nucleic Acids Res. 2016, 44(7), 3105-3117
    DOI: 10.1093/nar/gkv1372
  • Busch, T.; Draeger, G.; Kunst, E.; Benson, H.; Sasse, F.; Siems, K.; Kirschning, A. (2016): Synthesis and antiproliferative activity of new tonantzitlolone-derived diterpene derivatives.Org. Biomol. Chem. 2016, 14(38), 9040-9045
    DOI: 10.1039/c6ob01697a
  • Dibbert, N.; Krause, A.; Rios-Camacho, J.-C.; Gruh, I.; Kirschning, A.; Draeger, G. (2016): A Synthetic Toolbox for the In Situ Formation of Functionalized Homo- and Heteropolysaccharide-Based Hydrogel Libraries.Chem-Eur. J. 2016, 22(52), 18777-18786
    DOI: 10.1002/chem.201603748
  • Donner, J.; Reck, M.; Bergmann, S.; Kirschning, A.; Mueller, R.; Wagner-Doebler, I. (2016): The biofilm inhibitor Carolacton inhibits planktonic growth of virulent pneumococci via a conserved target.Scientific Reports 2016, 6
    DOI: 10.1038/srep29677
  • Gerstmann, L.; Kalesse, M. (2016): Total Synthesis of Aetheramide A.Chem-Eur. J. 2016, 22(32), 11210-11212
    DOI: 10.1002/chem.201602682
  • Gille, F.; Kirschning, A. (2016): Studies on the synthesis of peptides containing dehydrovaline and dehydroisoleucine based on copper-mediated enamide formation.Beilstein Journal of Organic Chemistry 2016, 12, 564-570
    DOI: 10.3762/bjoc.12.55
  • Graziadei, A.; Masiewicz, P.; Lapinaite, A.; Carlomagno, T. (2016): Archaea box C/D enzymes methylate two distinct substrate rRNA sequences with different efficiencyRNA. 2016, 22, 764-772
    DOI: 10.1261/rna.054320.115
  • Hartwig, J.; Kirschning, A. (2016): Flow Synthesis in Hot Water: Synthesis of the Atypical Antipsychotic Iloperidone.Chem-Eur J. 2016, 22(9), 3044-3052
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